The campaign
SHEET 01The published abstract, quoted
What happened, in five moves
SHEET 01Where this compound sits
SHEET 05The pocket
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Edit log
SHEET 03Contacts
SHEET 02Selected compound
SHEET 04Edit log
SHEET 03R-group grid
SHEET 04Activity cliffs
SHEET 04Compounds
SHEET 04Isoform selectivity
SHEET 04Potency against property
Ligand efficiency across the campaign
SHEET 05Pharmacokinetics by species
SHEET 05What you are looking at
SHEET 06The four papers are peer-reviewed work with Marc C. Deller as a co-author, contributing the protein crystallography. Every citation names all authors and links its DOI.